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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $24.65 | Total: $123.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 100 | $13.05 | Total: $1,305.00 |
Overview
NaV1.21.6 channel blocker-1 is a potent inhibitor of NaV1.2 and NaV1.6 channels, exhibiting inhibitory effects on rNaV1.6 and hNaV1.2. This compound can be utilized in the study of generalized epilepsy and movement disorders.
Chemical Properties
| Molecular Formula | C14H14N2OS |
| Molecular Weight | 258.34 |
| CAS Numbers | 1199944-04-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | S=C1OC=2C=CC=CC2C3=NC(=C(N13)CCC)C |
Storage and Handling
0C Short Term, -20C Long Term
References
Rivara M, et al. Biological Evaluation of Imidazobenzoxazines, Imidazobenzoxazin-5-ones and Imidazobenzoxazin-5-thiones as Sodium Channel Blockers. Letters in Drug Design & Discovery, 2014, 11, 90-97.