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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $67.15 | Total: $335.75 |
| 1 | 10 | $56.88 | Total: $568.80 |
| 1 | 25 | $48.19 | Total: $1,204.75 |
| 1 | 50 | $41.08 | Total: $2,054.00 |
| 1 | 100 | $35.55 | Total: $3,555.00 |
Overview
TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
Chemical Properties
| Molecular Formula | C13H12N2O4S |
| Molecular Weight | 292.31 |
| CAS Numbers | 2102179-29-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Oc1nc(sc1C(=O)N1CCCO1)-c1ccccc1O |
Storage and Handling
0C Short Term, -20C Long Term
References
Bianchini G, et al. Discovery of Novel TRPM8 Blockers Suitable for the Treatment of Somatic and Ocular Painful Conditions A Journey through pKa and LogD Modulation. J Med Chem. 2021 Nov 25;64[22] 16820-16837.