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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $24.65 | Total: $123.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 100 | $13.05 | Total: $1,305.00 |
Overview
PKM2-IN-1 (compound 3k) exhibits inhibitory activity against PKM2 with an IC50 of 2.95 ?M, while the IC50 for PKM1 is 4-5 times higher.
Chemical Properties
| Molecular Formula | C18H19NO2S2 |
| Molecular Weight | 345.48 |
| CAS Numbers | 94164-88-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC1=C(CSC(=S)N2CCCCC2)C(=O)c2ccccc2C1=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Ning X, et al. Discovery of novel naphthoquinone derivatives as inhibitors of the tumor cell specific M2 isoform of pyruvate kinase. Eur J Med Chem. 2017 Sep 29;138 343-352.
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