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NSC117079
AOB4882
CAS No: 500363-63-3
Chemical Name: NSC-117079; 1-Amino-9,10-dioxo-4-(3-sulfamoylanilino)anthracene-2-sulfonic acid
AOBIOUS launched this product in 2016
CITATIONS - Publications That Use AOBIOUS Product
310 Items
Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.95 | Total: $114.75 |
| 1 | 10 | $19.44 | Total: $194.40 |
| 1 | 25 | $16.47 | Total: $411.75 |
| 1 | 50 | $14.04 | Total: $702.00 |
| 1 | 100 | $12.15 | Total: $1,215.00 |
Overview
Novel pan-PHLPP inhibitors (selective for PHLPP1 and PHLPP2)
Chemical Properties
| Molecular Formula | C20H15N3O7S2 |
| Molecular Weight | 473.48 |
| CAS Numbers | 500363-63-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| IUPAC/Chemical Name | 1-Amino-9,10-dioxo-4-(3-sulfamoylanilino)anthracene-2-sulfonic acid |
| InChl Key | LHSBZAWDPSTOEY-UHFFFAOYSA-N |
| InChl Code | InChI=1S/C20H15N3O7S2/c21-18-15(32(28,29)30)9-14(23-10-4-3-5-11(8-10)31(22,26)27)16-17(18)20(25)13-7-2-1-6-12(13)19(16)24/h1-9,23H,21H2,(H2,22,26,27)(H,28,29,30) |
| SMILES Code | O=S(C(C(N)=C1C2=O)=CC(NC3=CC=CC(S(=O)(N)=O)=C3)=C1C(C4=C2C=CC=C4)=O)(O)=O |
Storage and Handling
0°C (short term), -20°C (long term), desiccated
Synonyms
NSC-117079; NSC 117079; NSC117079
References
1) Hwang SM, Feigenson M, Begun DL, Shull LC, Culley KL, Otero M, Goldring MB, Ta LE, Kakar S, Bradley EW, Westendorf JJ. Phlpp inhibitors block pain and cartilage degradation associated with osteoarthritis. J Orthop Res. 2018 May;36(5):1487-1497. doi: 10.1002/jor.23781. Epub 2017 Nov 28. PMID: 29068480; PMCID: PMC5985222.
2) Hwang SM, Feigenson M, Begun DL, Shull LC, Culley KL, Otero M, Goldring MB, Ta LE, Kakar S, Bradley EW, Westendorf JJ. Phlpp inhibitors block pain and cartilage degradation associated with osteoarthritis. J Orthop Res. 2018 May;36(5):1487-1497. doi: 10.1002/jor.23781. Epub 2017 Nov 28. PMID: 29068480; PMCID: PMC5985222.