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GKI-1
AOB8120
CAS No: 2444764-03-6
Chemical Name: Greatwall Kinase Inhibitor-1; N-(4-Chlorophenyl)-3-(1H-pyrazol-4-yl)aniline
926 Items
Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $31.45 | Total: $157.25 |
| 1 | 10 | $26.64 | Total: $266.40 |
| 1 | 25 | $22.57 | Total: $564.25 |
| 1 | 50 | $19.24 | Total: $962.00 |
| 1 | 100 | $16.65 | Total: $1,665.00 |
Overview
The first generation inhibitor of human Greatwall kinase, inhibiting full-length human GWL, and showing cellular efficacy
Chemical Properties
| Molecular Formula | C15H12ClN3 |
| Molecular Weight | 269.73 |
| CAS Numbers | 2444764-03-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| IUPAC/Chemical Name | N-(4-Chlorophenyl)-3-(1H-pyrazol-4-yl)aniline |
| SMILES Code | ClC(C=C1)=CC=C1NC2=CC(C3=CNN=C3)=CC=C2 |
Storage and Handling
0°C (short term), -20°C (long term), desiccated
Synonyms
Greatwall Kinase Inhibitor-1
References
1) Ocasio CA, et al. A first generation inhibitor of human Greatwall kinase, enabled by structural and functional characterisation of a minimal kinase domain construct. Oncotarget. 2016 Nov 1;7(44):71182-71197.
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