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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $23.80 | Total: $119.00 |
| 1 | 10 | $20.16 | Total: $201.60 |
| 1 | 25 | $17.08 | Total: $427.00 |
| 1 | 50 | $14.56 | Total: $728.00 |
| 1 | 100 | $12.60 | Total: $1,260.00 |
Overview
Pimitespib (TAS-116) is an ATP-competitive and highly specific HSP90?HSP90? inhibitor with inhibition constants (Kis) of 34.7 nM and 21.3 nM, respectively.
Chemical Properties
| Molecular Formula | C25H26N8O |
| Molecular Weight | 454.53 |
| CAS Numbers | 1260533-36-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCc1cc(ccc1-n1nc(C(C)C)c2c(ccnc12)-n1cnc(c1)-c1cnn(C)c1)C(N)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Ohkubo S, et al. TAS-116, a highly selective inhibitor of heat shock protein 90? and ?, demonstrates potent antitumor activity and minimal ocular toxicity in preclinical models. Mol Cancer Ther. 2015 Jan;14[1] 14-22.
