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Toll-Like Receptor (TLR)
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View larger TLR789-IN-1
AT39669
CAS 2180127-82-4
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $52.70 | Total: $263.50 |
| 1 | 10 | $44.64 | Total: $446.40 |
| 1 | 25 | $37.82 | Total: $945.50 |
| 1 | 50 | $32.24 | Total: $1,612.00 |
| 1 | 100 | $27.90 | Total: $2,790.00 |
Data sheet
| Molecular Formula | C27H37N3O2 |
| Molecular Weight | 435.6 |
| CAS Numbers | 2180127-82-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CNCCN1CCC(CC1)c1ccc2[nH]c(c(C(C)C)c2c1)-c1ccc(OC)c(OC)c1 |
| References | Mussari CP, et al. Discovery of Potent and Orally Bioavailable Small Molecule Antagonists of Toll-like Receptors 789 [TLR789]. ACS Med Chem Lett. 2020 Jul 29;11[9] 1751-1758. |
More info
TLR789-IN-1 is a potent inhibitor of Toll-like receptors 7, 8, and 9 (TLR789) with an IC50 of 43 nM.