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5HT Receptors
- Protein Control Ligand
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- Protease
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- Adenosine Deaminase
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- Cell Inhibition
- Synthase
- Receptor Tyrosine Phosphatases (RTP)
- AChE
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- Autophagy
- Toll-Like Receptor (TLR)
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- G Protein-Coupled Receptor Ligands
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- Adrenoceptor
- Angiotensin Receptor
- Cannabinoid Receptors
- CCK Receptors
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- EAA Receptors
- Ghrelin Receptors
- GABA Receptors
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- Metabotropic Glutamate Receptors
- Motilin Receptors
- Muscarinic Receptor
- Neuropeptide Receptors
- Opioid Receptors
- Orexin Receptors
- Orphan Receptors
- Prostanoid Receptors
- Proteinase-Activated Receptors
- Purinergic Receptors
- Ryanodine receptor
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- Thrombin Receptor
- Vaniloid Receptor
- VIP and PACAP Receptors
- Neurotensin Receptors
- Urotensin Receptor
- Imidazoline receptor
- SMO Receptors
- Apelin Receptor
- β-arrestin/β2-adaptin
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- Laminin Receptor
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- Amylin Receptor
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- CFTR
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- Biomarkers and Buffer Solutions
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View larger Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $13.05 | Total: $1,305.00 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 5 | $24.65 | Total: $123.25 |
Data sheet
| Molecular Formula | C18H15BrF2N4O2 |
| Molecular Weight | 437.24 |
| CAS Numbers | 839713-36-9 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1ccc(NC(=O)Nc2ccc(F)cc2F)cc1-c1c(Br)cnn1C |
| References | Al-Shamma H A , Anderson C , Chuang E , et al. Nelotanserin, a Novel Selective Human 5-Hydroxytryptamine2A Inverse Agonist for the Treatment of Insomnia[J]. Journal of Pharmacology and Experimental Therapeutics, 2010, 332[1] 281-290. |
More info
Nelotanserin (APD125) is a potent 5-HT2A inverse agonist(IC50 : 1.7 nM), a moderately potent 5-HT2C partial inverse agonist t(IC50 :79 nM )and a weak 5-HT2B inverse agonistt(IC50 : 791 nM).