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View larger Temanogrel
AT17033
CAS 887936-68-7
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $75.65 | Total: $378.25 |
| 1 | 10 | $64.08 | Total: $640.80 |
| 1 | 25 | $54.29 | Total: $1,357.25 |
| 1 | 50 | $46.28 | Total: $2,314.00 |
| 1 | 100 | $40.05 | Total: $4,005.00 |
Data sheet
| Molecular Formula | C24H28N4O4 |
| Molecular Weight | 436.5 |
| CAS Numbers | 887936-68-7 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1cccc(c1)C(=O)Nc1ccc(OCCN2CCOCC2)c(c1)-c1ccnn1C |
| References | Xiong Y, et al. Discovery and structure-activity relationship of 3-methoxy-N-[3-[1-methyl-1H-pyrazol-5-yl]-4-[2-morpholinoethoxy]phenyl]benzamide [APD791] a highly selective 5-hydroxytryptamine2A receptor inverse agonist for the treatment of arterial thrombosis. J Med Chem. 2010 Jun 10;53[11] 4412-21. |
More info
Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).