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> G Protein-Coupled Receptor Ligands>5HT Receptors>Naluzotan hydrochloride

5HT Receptors

Naluzotan hydrochloride View larger

Naluzotan hydrochloride

AT68113

CAS 740873-82-9

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$196.00

$196.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $166.60 Total: $833.00
110 $141.12 Total: $1,411.20
125 $119.56 Total: $2,989.00
150 $101.92 Total: $5,096.00
1100 $88.20 Total: $8,820.00

Data sheet

Molecular FormulaC23H39ClN4O3S
Molecular Weight487.1
CAS Numbers740873-82-9
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCl.O=C(NC1=CC=CC(=C1)N2CCN(CC2)CCCCNS(=O)(=O)CC3CCCCC3)C
ReferencesBecker OM, et al. An integrated in silico 3D model-driven discovery of a novel, potent, and selective amidosulfonamide 5-HT1A agonist [PRX-00023] for the treatment of anxiety and depression. J Med Chem. 2006 Jun 1;49[11] 3116-35.

More info

Naluzotan hydrochloride (PRX 00023 hydrochloride) is a hERG K+ channel blocker with an IC50 value of 3800 nM and is commonly used in the study of anxiety and depression.Naluzotan hydrochloride is also a novel, potent, and selective 5-HT1A agonist, with an IC50 value of about 20 nM and a Ki value of about 5.1 Naluzotan hydrochloride is also a novel, potent and selective 5-HT1A agonist with an IC50 of approximately 20 nM and a Ki of approximately 5.1 nM.