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View larger SB-616234-A
AT12847
CAS 908601-49-0
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $128.35 | Total: $641.75 |
| 1 | 10 | $108.72 | Total: $1,087.20 |
| 1 | 25 | $92.11 | Total: $2,302.75 |
| 1 | 50 | $78.52 | Total: $3,926.00 |
| 1 | 100 | $67.95 | Total: $6,795.00 |
Data sheet
| Molecular Formula | C32H36ClN5O3 |
| Molecular Weight | 574.11 |
| CAS Numbers | 908601-49-0 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.COc1cc2CCN(C(=O)c3ccc(cc3)-c3ccc(cc3C)-c3noc(C)n3)c2cc1N1C[C@H](C)N[C@H](C)C1 |
| References | Lee A.Dawson, et al. Characterisation of the selective 5-HT1B receptor antagonist SB-616234-A [1-[6-[cis-3,5-dimethylpiperazin-1-yl]-2,3-dihydro-5-methoxyindol-1-yl]-1-[2?-methyl-4?-[5-methyl-1,2,4-oxadiazol-3-yl]biphenyl-4-yl]methanone hydrochloride] In vivo neurochemical and behavioural evidence of anxiolyticantidepressant activity. Neuropharmacology Volume 50, Issue 8, June 2006, Pages 975-983 |
More info
SB-616234-A is a selective, orally bioavailable antagonist of the 5-HT1B receptor with anxiolytic and antidepressant properties.