5HT Receptors

NPS ALX Compound 4a hydrochloride(1:1) View larger

NPS ALX Compound 4a hydrochloride(1:1)

AT12262L1

Molarity Calculation Cart®

HOW TO ORDER

$71.00

$71.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $31.95 Total: $3,195.00
150 $36.92 Total: $1,846.00
125 $43.31 Total: $1,082.75
110 $51.12 Total: $511.20
15 $60.35 Total: $301.75

Data sheet

Molecular FormulaC25H26ClN3O2S
Molecular Weight468.01
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeO=S(C1=CC=CC2=C1C=CC=C2)(N3C=CC4=C3C=C(N5CCN6CCCC6C5)C=C4)=O.Cl
ReferencesIsaac M, et al. 6-Bicyclopiperazinyl-1-arylsulfonylindoles and 6-bicyclopiperidinyl-1-arylsulfonylindolesderivatives as novel, potent, and selective 5-HT6 receptor antagonists. Bioorg Med Chem Lett. 2000 Aug 7;10[15] 1719-21.

More info

NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM.