5HT Receptors

Didesmethyl cariprazine View larger

Didesmethyl cariprazine

AT15117

CAS 839712-25-3

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$126.00

$126.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $56.70 Total: $5,670.00
150 $65.52 Total: $3,276.00
125 $76.86 Total: $1,921.50
110 $90.72 Total: $907.20
15 $107.10 Total: $535.50

Data sheet

Molecular FormulaC19H28Cl2N4O
Molecular Weight399.36
CAS Numbers839712-25-3
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeNC(=O)N[C@H]1CC[C@H](CCN2CCN(CC2)c2cccc(Cl)c2Cl)CC1
ReferencesCitrome L, et al. Cariprazine for acute and maintenance treatment of adults with schizophrenia an evidence-based review and place in therapy. Neuropsychiatr Dis Treat. 2018;14 2563-2577.

More info

Didesmethyl cariprazine, a metabolite of Cariprazine, is the major cyclic active part. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a potent D3 preference D3D2 receptor partial agonist of dopamine for the treatment of schizophrenia, bipolar mania, and depression, with a high affinity for d3 and d2 receptors and a moderate affinity for 5-HT 1A receptors.