5HT Receptors

SB 258585 View larger

SB 258585

AT23318L

CAS 209480-63-7

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$35.00

$35.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $15.75 Total: $1,575.00
150 $18.20 Total: $910.00
125 $21.35 Total: $533.75
110 $25.20 Total: $252.00
15 $29.75 Total: $148.75

Data sheet

Molecular FormulaC18H22IN3O3S
Molecular Weight487.36
CAS Numbers209480-63-7
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeO=S(NC1=CC=C(C(N2CCN(CC2)C)=C1)OC)(C3=CC=C(C=C3)I)=O
ReferencesHirst WD, et al. Characterization of [[125]I]-SB-258585 binding to human recombinant and native 5-HT[6] receptors in rat, pig and human brain tissue. Br J Pharmacol. 2000 Aug;130[7] 1597-605.

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SB 258585 is a selective 5-HT6 receptor antagonist.SB 258585 has a high affinity for individual receptor populations in cell lines with human recombinant 5-HT6 receptors.SB 258585 can be used to label both recombinant and natural 5-HT6 receptors, and can be used to assay cognitive enhancement and antipsychotic activity.