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View larger Batefenterol
AT7079
CAS 743461-65-6
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $29.75 | Total: $148.75 |
| 1 | 10 | $25.20 | Total: $252.00 |
| 1 | 25 | $21.35 | Total: $533.75 |
| 1 | 50 | $18.20 | Total: $910.00 |
| 1 | 100 | $15.75 | Total: $1,575.00 |
Data sheet
| Molecular Formula | C40H42ClN5O7 |
| Molecular Weight | 740.24 |
| CAS Numbers | 743461-65-6 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1cc(NC(=O)CCN2CCC(CC2)OC(=O)Nc2ccccc2-c2ccccc2)c(Cl)cc1CNC[C@H](O)c1ccc(O)c2nc(O)ccc12 |
| References | Hegde SS, et al. Pharmacologic characterization of GSK-961081 [TD-5959], a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and ?2-adrenoceptor agonist properties. J Pharmacol Exp Ther. 2014 Oct;351[1] 190-9. |
More info
Batefenterol (TD-5959) (GSK961081, TD-5959) is a muscarinic receptor antagonist and ?2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic and h?2-adrenoceptor (Ki:1.41.33.7 nM).