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RO281675
AOB16496
CAS: 300352-96-9
Chemical Name: 3-Cyclopentyl-2-(4-(methylsulfonyl)phenyl)-N-(thiazol-2-yl)propanamide
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $8.55 | Total: $855.00 |
| 1 | 50 | $9.88 | Total: $494.00 |
| 1 | 25 | $11.59 | Total: $289.75 |
| 1 | 10 | $13.68 | Total: $136.80 |
| 1 | 5 | $16.15 | Total: $80.75 |
Data sheet
| Molecular Formula | C18H22N2O3S2 |
| Molecular Weight | 378.51 |
| CAS Numbers | 300352-96-9 |
| Storage Condition | 0°C (short term), -20°C (long term), desiccated |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| IUPAC/Chemical Name | 3-Cyclopentyl-2-(4-methanesulfonyl-phenyl)-N-thiazol-2-yl-propionamide |
| InChl Key | NEQSWPCDHDQINX-UHFFFAOYSA-N |
| InChl Code | InChI=1S/C18H22N2O3S2/c1-25(22,23)15-8-6-14(7-9-15)16(12-13-4-2-3-5-13)17(21)20-18-19-10-11-24-18/h6-11,13,16H,2-5,12H2,1H3,(H,19,20,21) |
| SMILES Code | CS(=O)(=O)C1=CC=C(C=C1)C(CC2CCCC2)C(=O)NC3=NC=CS3 |
| References | 1) Grimsby et al. Allosteric Activators of Glucokinase: Potential Role in Diabetes Therapy. Science Signaling 18 July 2003: 370. 2) T Kietzmann and GK Ganjam. Glucokinase: old enzyme, new target. Exp. Opin. Ther. Pat. 2005, 15, 705-713. |
More info
Novel glucokinase activator, selectively targeting L315H mutant and increasing insulin secretion