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View larger ADRA1D receptor antagonist 1 HCl
AT10250
CAS 1191908-14-1
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $76.05 | Total: $7,605.00 |
| 1 | 50 | $87.88 | Total: $4,394.00 |
| 1 | 25 | $103.09 | Total: $2,577.25 |
| 1 | 10 | $121.68 | Total: $1,216.80 |
| 1 | 5 | $143.65 | Total: $718.25 |
Data sheet
| Molecular Formula | C15H14Cl2N4O |
| Molecular Weight | 337.2 |
| CAS Numbers | 1191908-14-1 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.C[C@H](c1cccc(c1)C#N)n1cc(Cl)cc(C(N)=O)c1=N |
| References | Sakauchi N,et al. Discovery of 5-Chloro-1-[5-chloro-2-[methylsulfonyl]benzyl]-2-imino-1,2-dihydropyridine-3-carboxamide [TAK-259] as a Novel, Selective, and Orally Active ?1D Adrenoceptor Antagonist with Antiurinary Frequency Effects Reducing Human Ether-a-go-go-Related Gene [hERG] Liabilities. J Med Chem. 2016 Apr 14;59[7] 2989-3002. |
More info
ADRA1D receptor antagonist 1 HCl is an orally active, potent and selective ?1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activity.