Adrenoceptor

Saterinone View larger

Saterinone

AT68138

CAS 102669-89-6

More details

Molarity Calculation Cart®

HOW TO ORDER

$134.00

$134.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $60.30 Total: $6,030.00
150 $69.68 Total: $3,484.00
125 $81.74 Total: $2,043.50
110 $96.48 Total: $964.80
15 $113.90 Total: $569.50

Data sheet

Molecular FormulaC27H30N4O4
Molecular Weight474.55
CAS Numbers102669-89-6
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCC1=C(C=C(C#N)C(=O)N1)C2=CC=C(OCC(CN3CCN(CC3)C4=C(OC)C=CC=C4)O)C=C2
ReferencesBrunkhorst D, et al. Selective inhibition of cAMP phosphodiesterase III activity by the cardiotonic agent saterinone in guinea pig myocardium. Arzneimittelforschung. 1988;38[9] 1293-1298.

More info

Saterinone is a potent and selective phosphodiesterase III inhibitor and a potent antagonist of the vascular ?-1-adrenoceptor. Saterinone has vasodilatory properties and can be used in the acute treatment of chronic heart failure. Saterinone inhibited crude cAMP phosphodiesterase (PDE) activity in guinea pig right ventricular homogenates The ic50 value is 2.3