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> G Protein-Coupled Receptor Ligands>Adrenoceptor>G-Protein antagonist peptide acetate

Adrenoceptor

G-Protein antagonist peptide acetate View larger

G-Protein antagonist peptide acetate

ATP1902L1

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$118.00

$118.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $100.30 Total: $501.50
110 $84.96 Total: $849.60
125 $71.98 Total: $1,799.50
150 $61.36 Total: $3,068.00
1100 $53.10 Total: $5,310.00

Data sheet

Molecular FormulaC59H68N12O11S
Molecular Weight1153.33
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCSCC[C@@H](C(N)=O)NC([C@@H](CC1=CNC2=CC=CC=C12)NC([C@H](NC([C@H](CC3=CC=CC=C3)NC([C@H](NC([C@H](CCC(N)=O)NC([C@H]4NC(CC4)=O)=O)=O)CC5=CNC6=CC=CC=C56)=O)=O)CC7=CNC8=CC=CC=C78)=O)=O.CC(O)=O
ReferencesMukai H, et al. G protein antagonists. A novel hydrophobic peptide competes with receptor for G protein binding. J Biol Chem. 1992;267[23] 16237-16243.

More info

G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide acetate inhibits the activation of Gi or Go by M2 muscarinic cholinergic receptor (M2 mAChR) or of Gs by beta-adrenergic receptor in the reconstituted phospholipid vesicles, assayed by receptor-promoted GTP hydrolysis