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View larger BAY1082439
AT14511
CAS 1375469-38-7
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.10 | Total: $110.50 |
| 1 | 10 | $18.72 | Total: $187.20 |
| 1 | 25 | $15.86 | Total: $396.50 |
| 1 | 50 | $13.52 | Total: $676.00 |
| 1 | 100 | $11.70 | Total: $1,170.00 |
Data sheet
| Molecular Formula | C25H30N6O5 |
| Molecular Weight | 494.54 |
| CAS Numbers | 1375469-38-7 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1c(OC[C@H](O)CN2CCOCC2)ccc2C3=NCCN3C(NC(=O)c3cccnc3C)=Nc12 |
| References | Ningshu Liu, et al. Abstract 2799 BAY 1082439, a highly selective and balanced PI3K?? inhibitor demonstrated potent activity in tumors with activated PI3K? and loss-of-function of PTEN. Abstract nr 2799. doi 1538-7445.AM2012-2799. |
More info
BAY1082439, an orally bioavailable, selective inhibitor of PI3K???, demonstrates high efficacy in inhibiting the growth of Pten-null prostate cancer [1][2]. Additionally, BAY1082439 is effective against mutated forms of PIK3CA.