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> G Protein-Coupled Receptor Ligands>Bradykinin Receptor>R715 TFA(185052-09-9 free base)

Bradykinin Receptor

R715 TFA(185052-09-9 free base) View larger

R715 TFA(185052-09-9 free base)

ATP1933

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$129.00

$129.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $109.65 Total: $548.25
110 $92.88 Total: $928.80
125 $78.69 Total: $1,967.25
150 $67.08 Total: $3,354.00
1100 $58.05 Total: $5,805.00

Data sheet

Molecular FormulaC59H82F3N13O14
Molecular Weight1254.36
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCC[C@H](C)[C@@H](C(=O)O)NC(=O)[C@@H](CC1=CC2=CC=CC=C2C=C1)NC(=O)[C@H](CO)NC(=O)[C@H](CC3=CC=CC=C3)NC(=O)CNC(=O)[C@@H]4CCCN4C(=O)[C@@H]5CCCN5C(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCCN)NC(=O)C.OC(C(F)(F)F)=O
ReferencesGobeil et al [1996] Structure-activity studies of B1 receptor-related peptides. Hypertension. 28 833 PMID

More info

R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49). Displays no activity at B2 receptors. Reduces mechanical hypernociception in a mouse model of neuropathic pain. Metabolically stable.