Cannabinoid Receptors

Drinabant View larger

Drinabant

AT21861

CAS 358970-97-5

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$67.00

$67.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $30.15 Total: $3,015.00
150 $34.84 Total: $1,742.00
125 $40.87 Total: $1,021.75
110 $48.24 Total: $482.40
15 $56.95 Total: $284.75

Data sheet

Molecular FormulaC23H20Cl2F2N2O2S
Molecular Weight497.38
CAS Numbers358970-97-5
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeC(N1CC(N(S(C)(=O)=O)C2=CC(F)=CC(F)=C2)C1)(C3=CC=C(Cl)C=C3)C4=CC=C(Cl)C=C4
ReferencesAndreas W Herling, et al. CB1 receptor antagonist AVE1625 affects primarily metabolic parameters independently of reduced food intake in Wistar rats. Am J Physiol Endocrinol Metab. 2007 Sep;293[3] E826-32.

More info

Drinabant (AVE-1625) is an orally active CB1 receptor antagonist. Drinabant inhibits the agonist-stimulated calcium signal with IC50 values of 25 nM and 10 nM for the hCB1-R and rCB1-R, respectively, and is ineffective for the hCB2-R.