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CGRP Receptor
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View larger CGRP antagonist 1
AT13453
CAS 1123757-49-2
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $247.35 | Total: $1,236.75 |
| 1 | 10 | $209.52 | Total: $2,095.20 |
| 1 | 25 | $177.51 | Total: $4,437.75 |
| 1 | 50 | $151.32 | Total: $7,566.00 |
| 1 | 100 | $130.95 | Total: $13,095.00 |
Data sheet
| Molecular Formula | C29H26N4O4 |
| Molecular Weight | 494.54 |
| CAS Numbers | 1123757-49-2 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C1[C@]2(C=3C(N1)=NC=CC3)CC=4C(C2)=CC=C(NC(CN5C=6C(C7(C5=O)CCOCC7)=CC=CC6)=O)C4 |
| References | Stump CA, et al. The discovery of highly potent CGRP receptor antagonists. Bioorg Med Chem Lett. 2009 Jan 1;19[1] 214-7. |
More info
CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the study of cardiovascular and neurovascular diseases.