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BM221
AOB12963
CAS N/A
Chemical Name: Ac-Phe-Lys-Pro-Leu-Ala-Abu-D-Ala-Arg-OH
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HOW TO ORDER
Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $58.05 | Total: $5,805.00 |
| 1 | 50 | $67.08 | Total: $3,354.00 |
| 1 | 25 | $78.69 | Total: $1,967.25 |
| 1 | 10 | $92.88 | Total: $928.80 |
| 1 | 5 | $109.65 | Total: $548.25 |
Data sheet
| Molecular Formula | C44H72N12O10 |
| Molecular Weight | 929.13 |
| Storage Condition | 0°C (short term), -20°C (long term), desiccated |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| Synonym | BM221; BM 221; BM-221 |
| IUPAC/Chemical Name | ((S)-2-((S)-2-((S)-2-((S)-1-(acetyl-L-phenylalanyl-L-lysyl)pyrrolidine-2-carboxamido)-4-methylpentanamido)propanamido)butanoyl)-D-alanyl-L-arginine |
| InChl Key | XDOOBNYHWWUCRX-ZNLDZGKTSA-N |
| InChl Code | InChI=1S/C44H72N12O10/c1-7-30(38(60)49-27(5)37(59)54-32(43(65)66)18-13-21-48-44(46)47)52-36(58)26(4)50-39(61)33(23-25(2)3)55-41(63)35-19-14-22-56(35)42(64)31(17-11-12-20-45)53-40(62)34(51-28(6)57)24-29-15-9-8-10-16-29/h8-10,15-16,25-27,30-35H,7,11-14,17-24,45H2,1-6H3,(H,49,60)(H,50,61)(H,51,57)(H,52,58)(H,53,62)(H,54,59)(H,55,63)(H,65,66)(H4,46,47,48)/t26-,27+,30-,31-,32-,33-,34-,35-/m0/s1 |
| SMILES Code | O=C(N[C@@H](CC1=CC=CC=C1)C(N[C@@H](CCCCN)C(N2[C@@H](CCC2)C(N[C@@H](CC(C)C)C(N[C@@H](C)C(N[C@@H](CC)C(N[C@H](C)C(N[C@@H](CCCNC(N)=N)C(O)=O)=O)=O)=O)=O)=O)=O)=O)C |
| References | 1) Gorman DM, Li XX, Lee JD, Fung JN, Cui CS, Lee HS, Rolfe BE, Woodruff TM, Clark RJ. Development of Potent and Selective Agonists for Complement C5a Receptor 1 with In Vivo Activity. J Med Chem. 2021 Nov 25;64(22):16598-16608. doi: 10.1021/acs.jmedchem.1c01174. Epub 2021 Nov 11. PMID: 34762432. |
More info
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