EAA Receptors

Flupirtine Maleate View larger

Flupirtine Maleate

AOB0383

 

CAS No: 75507-68-5

 

Chemical Name: Katadolon; Ethyl N-[2-amino-6-[(4-fluorophenyl)methylamino]pyridin-3-yl]carbamate Maleate

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Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $4.05 Total: $405.00
150 $4.68 Total: $234.00
125 $5.49 Total: $137.25
110 $6.48 Total: $64.80
15 $7.65 Total: $38.25

Data sheet

Molecular FormulaC19H21FN4O6
Molecular Weight420.39
CAS Numbers75507-68-5
Storage Condition0°C (short term), -20°C (long term), desiccated
SolubilityDMSO
Purity98% by HPLC
SynonymFlupirtine; W-2964M; W2964M; W 2964M; W-2964; W2964; W 2964; D-9998; Katadolon.
IUPAC/Chemical Nameethyl (2-amino-6-((4-fluorobenzyl)amino)pyridin-3-yl)carbamate maleate
InChl Keyethyl (2-amino-6-((4-fluorobenzyl)amino)pyridin-3-yl)carbamate maleate
InChl CodeInChI=1S/C15H17FN4O2.C4H4O4/c1-2-22-15(21)19-12-7-8-13(20-14(12)17)18-9-10-3-5-11(16)6-4-10;5-3(6)1-2-4(7)8/h3-8H,2,9H2,1H3,(H,19,21)(H3,17,18,20);1-2H,(H,5,6)(H,7,8)/b;2-1-
SMILES CodeO=C(OCC)NC1=CC=C(NCC2=CC=C(F)C=C2)N=C1N.O=C(O)/C=CC(O)=O
References1) Wörz R. [Long-term-treatment of chronic pain patients with flupirtine--on hepatotoxicity and persistent effectiveness from 7 months to 22 years]. MMW Fortschr Med. 2014 Dec 15;156 Suppl 4:127-34. Review. German. PubMed PMID: 26153592.

2) Szelenyi I. Flupirtine, a re-discovered drug, revisited. Inflamm Res. 2013 Mar;62(3):251-8.
PubChem ID53276

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