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View larger Methoxy-PEPy
AT12012
CAS 524924-76-3
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.10 | Total: $110.50 |
| 1 | 10 | $18.72 | Total: $187.20 |
| 1 | 25 | $15.86 | Total: $396.50 |
| 1 | 50 | $13.52 | Total: $676.00 |
| 1 | 100 | $11.70 | Total: $1,170.00 |
Data sheet
| Molecular Formula | C13H10N2O |
| Molecular Weight | 210.23 |
| CAS Numbers | 524924-76-3 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1cncc(c1)C#Cc1ccccn1 |
| References | Cosford ND, et al. [3H]-methoxymethyl-MTEP and [3H]-methoxy-PEPy potent and selective radioligands for the metabotropic glutamate subtype 5 [mGlu5] receptor. Bioorg Med Chem Lett. 2003 Feb 10;13[3] 351-4. |
More info
Methoxy-PEPy is a potent and selective mGlu5 receptor inhibitor, exhibiting an IC50 value of 1 nM.