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View larger CCG-257081
AT30778
CAS 1922098-90-5
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $93.50 | Total: $467.50 |
| 1 | 10 | $79.20 | Total: $792.00 |
| 1 | 25 | $67.10 | Total: $1,677.50 |
| 1 | 50 | $57.20 | Total: $2,860.00 |
| 1 | 100 | $49.50 | Total: $4,950.00 |
Data sheet
| Molecular Formula | C24H19ClF3N3O2 |
| Molecular Weight | 473.87 |
| CAS Numbers | 1922098-90-5 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(=O)(C=1C=C(C=C(F)C1)C=2C=CN=CC2)N3CC(C(NC4=CC=C(Cl)C=C4)=O)CC(F)(F)C3 |
| References | Larsen Scott D, et al. Preparation of substituted piperidine-3-carboxamides as inhibitors of myocardin-related transcription factor and serum response factor [MTRFSRF]-mediated gene transcription. WO2016073847 A2. |
More info
CCG-257081 (MRTFSRF-IN-1) is an inhibitor of cardiac myosin-related transcription factor and serum response factor (MRTFSRF) that acts by inhibiting the RhoMRTFSRF pathway.CCG-257081 has shown efficacy in preventing bleomycin-induced fibrosis in several mouse models. CCG-257081 can be used in cancer prevention and fibrosis research.