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View larger Ruboxistaurin hydrochloride
AT3689
CAS 169939-93-9
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $46.75 | Total: $233.75 |
| 1 | 10 | $39.60 | Total: $396.00 |
| 1 | 25 | $33.55 | Total: $838.75 |
| 1 | 50 | $28.60 | Total: $1,430.00 |
| 1 | 100 | $24.75 | Total: $2,475.00 |
Data sheet
| Molecular Formula | C28H28N4O3 |
| Molecular Weight | 505.01 |
| CAS Numbers | 169939-93-9 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.CN(C)CC1CCn2cc(C3=C(C(=O)NC3=O)c3cn(CCO1)c1ccccc31)c1ccccc21 |
| References | Jirousek MR, et al. J Med Chem. 1996, 39[14] 2664-71. |
More info
Ruboxistaurin hydrochloride (LY 333531 hydrochloride) is an Isozyme-selective inhibitor of protein kinase C (PKC); competitively and reversibly inhibits PKC?I and PKC?II (IC50 values are 4.7 and 5.9 nM respectively). Selective for PKC? over other PKC isozymes (IC50values are 0.052, 0.25, 0.30, 0.36, 0.60 and >100 ?M for PKC?, -?, -?, -?, -? and -? respectively). Exhibits selectivity for PKC over other ATP-dependent kinases, including protein kinase A, casein kinase and src).