> Pathway Inhibitors>Enzyme Inhibitors>PKA Inhibitor Fragment (6-22) amide TFA

Enzyme Inhibitors

PKA Inhibitor Fragment (6-22) amide TFA View larger

PKA Inhibitor Fragment (6-22) amide TFA

AT75888

Molarity Calculation Cart®

HOW TO ORDER

$127.00

$127.00 per mg

Add to my wishlist

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $57.15 Total: $5,715.00
150 $66.04 Total: $3,302.00
125 $77.47 Total: $1,936.75
110 $91.44 Total: $914.40
15 $107.95 Total: $539.75

Data sheet

Molecular FormulaC82H131F3N28O26
Molecular Weight1982.08
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCC[C@H](C)[C@@H](C(N)=O)NC([C@H](C)NC([C@H](CC(N)=O)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC(CNC([C@H]([C@H](O)C)NC([C@H](CCCNC(N)=N)NC(CNC([C@H](CO)NC([C@H](C)NC([C@H]([C@@H](C)CC)NC([C@@H](NC([C@H](CC(O)=O)NC([C@H](C)NC([C@@H](NC([C@@H](N)[C@H](O)C)=O)CC1=CC=C(C=C1)O)=O)=O)=O)CC2=CC=CC=C2)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O.OC(C(F)(F)F)=O
ReferencesDalton GD, et al. Alterations in brain Protein Kinase A activity and reversal of morphine tolerance by two fragments of native Protein Kinase A inhibitor peptide [PKI]. Neuropharmacology. 2005 Apr; 48[5] 648-57.

More info

PKA Inhibitor Fragment (6-22) amide TFA (PKA Inhibitor Fragment (6-22) amide TFA) is a highly potent inhibitor of cAMP-dependent protein kinase A (PKA) with a Ki of 2.8 nM and reverses the pain-relieving effects of low levels of morphine in mice.