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View larger Rilapladib
AT16751
CAS 412950-08-4
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $68.00 | Total: $340.00 |
| 1 | 10 | $57.60 | Total: $576.00 |
| 1 | 25 | $48.80 | Total: $1,220.00 |
| 1 | 50 | $41.60 | Total: $2,080.00 |
| 1 | 100 | $36.00 | Total: $3,600.00 |
Data sheet
| Molecular Formula | C40H38F5N3O3S |
| Molecular Weight | 735.8 |
| CAS Numbers | 412950-08-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COCCN1CCC(CC1)N(Cc1ccc(cc1)-c1ccc(cc1)C(F)(F)F)C(=O)Cn1c(SCc2cccc(F)c2F)cc(=O)c2ccccc12 |
| References | Shaddinger BC, et al. Platelet aggregation unchanged by lipoprotein-associated phospholipase A? inhibition results from an in vitro study and two randomized phase I trials. PLoS One. 2014 Jan 27;9[1] e83094. |
More info
Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA2, IC50 = 230 pM) and acts as an antagonist of the platelet-activating factor receptor.