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Enzyme Inhibitors
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View larger Tafetinib
AT28911
CAS 1032265-57-8
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $181.05 | Total: $905.25 |
| 1 | 10 | $153.36 | Total: $1,533.60 |
| 1 | 25 | $129.93 | Total: $3,248.25 |
| 1 | 50 | $110.76 | Total: $5,538.00 |
| 1 | 100 | $95.85 | Total: $9,585.00 |
Data sheet
| Molecular Formula | C24H29FN4O2 |
| Molecular Weight | 424.51 |
| CAS Numbers | 1032265-57-8 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C1C(=C2C3=C(C(C(NCCN(CC)CC)=O)=C(C)N3)CCC2)C=4C(N1)=CC=C(F)C4 |
| References | Shao F, et al. Simultaneous quantification of tafetinib [SIM010603], a novel potent inhibitor of receptor tyrosine kinase, and its major metabolite in dog plasma by HPLC-ESIMSMS and its application to a pharmacokinetic study. J Pharm Biomed Anal. 2013 Jul-Aug;81-82 50-5. |
More info
Tafetinib (SIM-010603) is a novel potent and orally available tyrosine kinase inhibitor with anti-angiogenic and anti-tumour activity.