Enzyme Inhibitors

YAP-TEAD-IN-1 acetate View larger

YAP-TEAD-IN-1 acetate

ATP2160L1

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HOW TO ORDER

$125.00

$125.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $56.25 Total: $5,625.00
150 $65.00 Total: $3,250.00
125 $76.25 Total: $1,906.25
110 $90.00 Total: $900.00
15 $106.25 Total: $531.25

Data sheet

Molecular FormulaC95H148ClN23O23S2
Molecular Weight2079.92
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeO=C(N(CCC1)[C@@H]1C(N[C@@H](C(N)=O)CCC(O)=O)=O)[C@H](CCC2)N2C([C@H](CCCCN)NC([C@H](CSSCC[C@@H](C(N[C@H](C(N[C@@H](C(N[C@H]3CCCCN)=O)CCCNC(N)=N)=O)CC(C)C)=O)NC([C@H](CC4=CC(Cl)=CC=C4)NC([C@H](CCC5)N5C([C@H](C(C)C)NC(C)=O)=O)=O)=O)NC([C@@H](NC([C@@](NC([C@@H](NC([C@@](CCC6)([H])N6C([C@](NC3=O)([H])CCCC)=O)=O)C)=O)([H])CO)=O)CC7=CC=CC=C7)=O)=O)=O.CC(O)=O
ReferencesZhang Z, et al. Structure-Based Design and Synthesis of Potent Cyclic Peptides Inhibiting the YAP-TEAD Protein-Protein Interaction.ACS Med Chem Lett. 2014 Jul 14;5[9] 993-8.

More info

YAP-TEAD-IN-1 acetate is an effective and competitive inhibitor of YAP