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Enzyme Inhibitors
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View larger CPI-0610 carboxylic acid
AT10879
CAS 1380089-81-5
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $379.95 | Total: $1,899.75 |
| 1 | 10 | $321.84 | Total: $3,218.40 |
| 1 | 25 | $272.67 | Total: $6,816.75 |
| 1 | 50 | $232.44 | Total: $11,622.00 |
| 1 | 100 | $201.15 | Total: $20,115.00 |
Data sheet
| Molecular Formula | C20H15ClN2O3 |
| Molecular Weight | 366.8 |
| CAS Numbers | 1380089-81-5 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC=1C=2C=3C(C(=N[C@@H](CC(O)=O)C2ON1)C4=CC=C(Cl)C=C4)=CC=CC3 |
| References | Albrecht BK, et al. Identification of a Benzoisoxazoloazepine Inhibitor [CPI-0610] of the Bromodomain and Extra-Terminal [BET] Family as a Candidate for Human Clinical Trials. J Med Chem. 2016;59[4] 1330-1339. |
More info
CPI-0610 carboxylic acid is an effective and selective small molecule inhibitor of bromine domain and outer end (BET) protein as a ligand of PROTAC target protein. CPI-0610 carboxylic acid may have anticancer and anticancer activities.