Enzyme Inhibitors

LY2955303 View larger

LY2955303

AT15811

CAS 1433497-19-8

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$30.00

$30.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $13.50 Total: $1,350.00
150 $15.60 Total: $780.00
125 $18.30 Total: $457.50
110 $21.60 Total: $216.00
15 $25.50 Total: $127.50

Data sheet

Molecular FormulaC36H42N4O3
Molecular Weight578.74
CAS Numbers1433497-19-8
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCN1CCN(CC1)C(=O)c1ccc(cc1)-n1nc(cc1-c1cc(cc(c1)C(C)(C)C)C(C)(C)C)-c1ccc(cc1)C(O)=O
ReferencesHughes NE, et al. Identification of potent and selective retinoic acid receptor gamma [RAR?] antagonists for the treatment of osteoarthritis pain using structure based drug design. Bioorg Med Chem Lett. 2016 Jul 15;26[14] 3274-3277.

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LY2955303 is an effective and selective antagonist of retinoic acid receptor gamma (RAR?, Ki = 1.09 nM).