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View larger AHR antagonist 5 free base
AT39762
CAS 2247950-42-9
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $112.20 | Total: $561.00 |
| 1 | 10 | $95.04 | Total: $950.40 |
| 1 | 25 | $80.52 | Total: $2,013.00 |
| 1 | 50 | $68.64 | Total: $3,432.00 |
| 1 | 100 | $59.40 | Total: $5,940.00 |
Data sheet
| Molecular Formula | C25H24FN7 |
| Molecular Weight | 441.5 |
| CAS Numbers | 2247950-42-9 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(C=1N2C(=C(C(C)C)C=N2)N=C(N1)C=3C=C(F)C=NC3)[C@H]4CC=5C=6C(NC5CC4)=CC=CC6 |
| References | Marta Sanchez-Martin, et al. Ahr inhibitors and uses thereof. WO2021142180A1. |
More info
AHR antagonist 5 free base is an orally active antagonist of AHR with IC50s of approximately 35-150 nM in human and rodent cell lines (in vitro).