Epigenetics

SR 16832 View larger

SR 16832

AT24827

CAS 2088135-12-8

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$26.00

$26.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $11.70 Total: $1,170.00
150 $13.52 Total: $676.00
125 $15.86 Total: $396.50
110 $18.72 Total: $187.20
15 $22.10 Total: $110.50

Data sheet

Molecular FormulaC17H12ClN3O4
Molecular Weight357.75
CAS Numbers2088135-12-8
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeN(C(=O)C1=CC(N(=O)=O)=CC=C1Cl)C=2C3=C(C=CC(OC)=C3)N=CC2
ReferencesBrust et al [2017] Modification of the othosteric PPAR? covalent antagonist scaffold yields an improved dual-site allosteric inhibitor. ACS Chem.Biol. 12 969

More info

SR 16832 is a dual-site PPAR? inhibitor. It also inhibits the binding of endogenous ligands and transcriptional activity of PPAR?, more effectively than the orthosteric covalent antagonist GW 9662 and T 0070907.