Epigenetics

ZEN-3862 View larger

ZEN-3862

AT13394

CAS 1952264-33-3

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$49.00

$49.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $22.05 Total: $2,205.00
150 $25.48 Total: $1,274.00
125 $29.89 Total: $747.25
110 $35.28 Total: $352.80
15 $41.65 Total: $208.25

Data sheet

Molecular FormulaC19H17FN2O3
Molecular Weight340.35
CAS Numbers1952264-33-3
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCC=1C(C2=CN(CC3=CC(F)=C(C=C3)C4CO4)C(=O)C=C2)=C(C)ON1
ReferencesKharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain [BET] Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61[18] 8202-8211.

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ZEN-3862 (Willardiine) is an inhibitor of BET(IC50s of 0.16 and 0.13 ?M for BRD4(BD1) and BRD4(BD2) , respectively). ZEN-3862 can be used to form PROTACs to induce degradation of BRD4.