Epigenetics

ZEN-3411 View larger

ZEN-3411

AT13393

CAS 1952264-36-6

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$298.00

$298.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $134.10 Total: $13,410.00
150 $154.96 Total: $7,748.00
125 $181.78 Total: $4,544.50
110 $214.56 Total: $2,145.60
15 $253.30 Total: $1,266.50

Data sheet

Molecular FormulaC21H20N4O2
Molecular Weight360.41
CAS Numbers1952264-36-6
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeC(N1C=2C(=C(N)C=C(C2)C=3C(C)=NOC3C)N=C1)C4=CC=C(C=C4)C5CO5
ReferencesKharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain [BET] Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61[18] 8202-8211.

More info

ZEN-3411 is an orally available and potent BET inhibitor that inhibits BRD4(BD1), BRD4(BD2), and BRD4(BD1BD2) and suppresses the growth of tumor cells overproducing BET proteins.