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View larger KDM5-IN-1
AT15649
CAS 1628210-26-3
1000 Items
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $41.65 | Total: $208.25 |
| 1 | 10 | $35.28 | Total: $352.80 |
| 1 | 25 | $29.89 | Total: $747.25 |
| 1 | 50 | $25.48 | Total: $1,274.00 |
| 1 | 100 | $22.05 | Total: $2,205.00 |
Data sheet
| Molecular Formula | C17H20N6O |
| Molecular Weight | 324.38 |
| CAS Numbers | 1628210-26-3 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(C)c1c([nH]c2c(cnn2c1=O)C#N)-c1cnn(c1)C(C)(C)C |
| References | Liang J, et al. Lead optimization of a pyrazolo[1,5-a]pyrimidin-7[4H]-one scaffold to identify potent, selective and orally bioavailable KDM5 inhibitors suitable for in vivo biological studies. Bioorg Med Chem Lett. 2016 Aug 15;26[16] 4036-41. |
More info
KDM5-IN-1 is an effective and selective inhibitor of KDM5 with an IC50 of 15.1 nM.