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Epigenetics
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View larger DC-BPi-03
AT73288
CAS 2758411-46-8
1000 Items
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $160.65 | Total: $803.25 |
| 1 | 10 | $136.08 | Total: $1,360.80 |
| 1 | 25 | $115.29 | Total: $2,882.25 |
| 1 | 50 | $98.28 | Total: $4,914.00 |
| 1 | 100 | $85.05 | Total: $8,505.00 |
Data sheet
| Molecular Formula | C14H14N4O2S |
| Molecular Weight | 302.35 |
| CAS Numbers | 2758411-46-8 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=S(=O)(C=1N=C(C=C(N1)C2=CC=C3NC=CC3=C2)NC)C |
| References | Tian Lu, et al. Discovery of High-Affinity Inhibitors of the BPTF Bromodomain. J Med Chem. 2021 Aug 26;64[16] 12075-12088. |
More info
DC-BPi-03 is a potent BPTF-BRD inhibitor, exhibiting an IC50 of 698.3 nM and a Kd of 2.81 ?M.