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AP1189
AOB31893
CAS: 959850-74-9
Chemical Name: (E)-N-[trans-3-{1-(2-Nitrophenyl)-1H-pyrrol-2-yl} allylidenamino]guanidinium acetate
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity (mg or Unit) | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|
| 100 | $9.45 | Total: $945.00 |
| 50 | $10.92 | Total: $546.00 |
| 25 | $12.81 | Total: $320.25 |
| 10 | $15.12 | Total: $151.20 |
| 5 | $17.85 | Total: $89.25 |
Data sheet
| Molecular Formula | C16H18N6O4 |
| Molecular Weight | 358.36 |
| CAS Numbers | 959850-74-9 |
| Storage Condition | 0°C (short term), -20°C (long term), desiccated |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| Synonym | AP-1189; AP 1189; AP1189; AP1189 acetate; |
| IUPAC/Chemical Name | (E)-N-[trans-3-{1-(2-Nitrophenyl)-1H-pyrrol-2-yl} allylidenamino]guanidinium acetate |
| InChl Key | FIESOFUABUPMMH-WAJHRQJSSA-N |
| InChl Code | InChI=1S/C14H14N6O2.C2H4O2/c15-14(16)18-17-9-3-5-11-6-4-10-19(11)12-7-1-2-8-13(12)20(21)22;1-2(3)4/h1-10H,(H4,15,16,18);1H3,(H,3,4)/b5-3+,17-9+; |
| SMILES Code | NC(N/N=C/C=C/C1=CC=CN1C2=CC=CC=C2[N+]([O-])=O)=N.CC(O)=O |
| References | 1) Montero-Melendez T, Gobbetti T, Cooray SN, Jonassen TE, Perretti M. Biased agonism as a novel strategy to harness the proresolving properties of melanocortin receptors without eliciting melanogenic effects. J Immunol. 2015 Apr 1;194(7):3381-8. doi: 10.4049/jimmunol.1402645. Epub 2015 Feb 27. PubMed PMID: 25725103. |
More info
Novel biased agonist at receptors MC1 and MC3