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> G Protein-Coupled Receptor Ligands>d[Leu4,Lys8]-VP acetate

G Protein-Coupled Receptor Ligands

d[Leu4,Lys8]-VP acetate View larger

d[Leu4,Lys8]-VP acetate

ATP1927L1

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$33.00

$33.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $28.05 Total: $140.25
110 $23.76 Total: $237.60
125 $20.13 Total: $503.25
150 $17.16 Total: $858.00
1100 $14.85 Total: $1,485.00

Data sheet

Molecular FormulaC49H71N11O13S2
Molecular Weight1086.28
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCC(O)=O.NC(CNC([C@@H](NC([C@@H]1CCCN1C([C@@H](NC([C@@H]2CC(N)=O)=O)CSSCCC(N[C@H](C(N[C@](CC3=CC=CC=C3)([H])C(N[C@@H](CC(C)C)C(N2)=O)=O)=O)CC4=CC=C(O)C=C4)=O)=O)=O)CCCCN)=O)=O
ReferencesAna P, et, al. Design and synthesis of the first selective agonists for the rat vasopressin V[1b] receptor based on modifications of deamino-[Cys1]arginine vasopressin at positions 4 and 8. J Med Chem. 2007 Feb 22; 50[4] 835-47.

More info

d[Leu4,Lys8]-VP acetate is a selective vasopressin V1b receptor agonist. The Kis for rat, human and mouse V1b receptors are 0.16 nM, 0.52 nM and 0.1.38 nM, respectively. d[Leu4,Lys8]-VP acetate exhibits weak antidiuretic, vasopressor and oxytocic activiti