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> G Protein-Coupled Receptor Ligands>PG 106 acetate

G Protein-Coupled Receptor Ligands

PG 106 acetate View larger

PG 106 acetate

ATP1952L

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$150.00

$150.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $127.50 Total: $637.50
110 $108.00 Total: $1,080.00
125 $91.50 Total: $2,287.50
150 $78.00 Total: $3,900.00
1100 $67.50 Total: $6,750.00

Data sheet

Molecular FormulaC53H73N13O11
Molecular Weight1068.23
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCCCCC(NC(C)=O)C(N[C@H]1CC(NCCCC[C@@H](C(N)=O)NC([C@H](CC2=CNC3=CC=CC=C32)NC([C@H](CCCN=C(N)N)NC([C@@H](CC4=CC5=CC=CC=C5C=C4)NC(CCNC1=O)=O)=O)=O)=O)=O)=O.CC(O)=O
ReferencesPaolo Grieco, et al. Further structure-activity studies of lactam derivatives of MT-II and SHU-9119 their activity and selectivity at human melanocortin receptors 3, 4, and 5. Peptides

More info

PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM.