G Protein-Coupled Receptor Ligands

TASP0390325 View larger

TASP0390325

AT28926

CAS 1642187-96-9

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$44.00

$44.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $19.80 Total: $1,980.00
150 $22.88 Total: $1,144.00
125 $26.84 Total: $671.00
110 $31.68 Total: $316.80
15 $37.40 Total: $187.00

Data sheet

Molecular FormulaC25H30Cl2FN5O4
Molecular Weight554.44
CAS Numbers1642187-96-9
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCl.O=C1C2=CC(OCCCN3CCOCC3)=CN=C2N=C(C=4C=CC(F)=C(Cl)C4)N1CC(=O)NC(C)C
ReferencesM Iijima, et al. Antidepressant and anxiolytic profiles of newly synthesized arginine vasopressin V1B receptor antagonists TASP0233278 and TASP0390325. Br J Pharmacol. 2014 Jul;171[14] 3511-25.

More info

TASP0390325 is an orally active and high affinity arginine pressin receptor 1B (V1B receptor) antagonist that shows antidepressant and anxiolytic activity in animal studies and blocks V1B receptors in the anterior pituitary gland in vivo.