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View larger TG 100572 Hydrochloride
AT13156L
CAS 867331-64-4
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $288.15 | Total: $1,440.75 |
| 1 | 10 | $244.08 | Total: $2,440.80 |
| 1 | 25 | $206.79 | Total: $5,169.75 |
| 1 | 50 | $176.28 | Total: $8,814.00 |
| 1 | 100 | $152.55 | Total: $15,255.00 |
Data sheet
| Molecular Formula | C26H27Cl2N5O2 |
| Molecular Weight | 512.43 |
| CAS Numbers | 867331-64-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.Cc1cc(cc2nnc(Nc3ccc(OCCN4CCCC4)cc3)nc12)-c1cc(O)ccc1Cl |
| References | Doukas J, et al. Topical administration of a multi-targeted kinase inhibitor suppresses choroidal neovascularization and retinal edema. J Cell Physiol. 2008 Jul;216[1] 29-37. |
More info
TG 100572 Hydrochloride is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src kinases(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 nM for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFR?, Fgr, Fyn, Hck, Lck, Lyn, Src, Yes, respectively).