G Protein-Coupled Receptor Ligands

d[Cha4]-AVP acetate(500170-27-4 free base) View larger

d[Cha4]-AVP acetate(500170-27-4 free base)

ATP2082L

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$85.00

$85.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $38.25 Total: $3,825.00
150 $44.20 Total: $2,210.00
125 $51.85 Total: $1,296.25
110 $61.20 Total: $612.00
15 $72.25 Total: $361.25

Data sheet

Molecular FormulaC52H75N13O13S2
Molecular Weight1154.37
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeO=C(N[C@@H](CC(N)=O)C(N[C@H](C(N1CCC[C@H]1C(N[C@H](C(NCC(N)=O)=O)CCCN=C(N)N)=O)=O)CSSCCC(N[C@@H](CC2=CC=C(O)C=C2)C(N[C@@H](CC3=CC=CC=C3)C(N4)=O)=O)=O)=O)[C@@H]4CC5CCCCC5.CC(O)=O
ReferencesDerick et al [2002] [1-Deamino-4-cyclohexylalanine] arginine vasopressin a potent and specific agonist for vasopressin V1b receptors. Endocrinology 143 4655 PMID

More info

d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively). Stimulates ACTH and corticosterone secretion and exhibits negligible vasopressor activity in vivo.