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View larger (E)-GABAB receptor antagonist 1
AT11137
CAS 1611483-29-4
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $74.70 | Total: $7,470.00 |
| 1 | 50 | $86.32 | Total: $4,316.00 |
| 1 | 25 | $101.26 | Total: $2,531.50 |
| 1 | 10 | $119.52 | Total: $1,195.20 |
| 1 | 5 | $141.10 | Total: $705.50 |
Data sheet
| Molecular Formula | C18H24O4 |
| Molecular Weight | 304.38 |
| CAS Numbers | 1611483-29-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(=CC(C(O)=O)=O)C1=CC(C(C)(C)C)=C(O)C(C(C)(C)C)=C1 |
| References | Chen LH, et al. Discovery of a Negative Allosteric Modulator of GABAB Receptors. ACS Med Chem Lett. 2014 May 27;5[7] 742-7. |
More info
(E)-GABAB receptor antagonist 1 is a trans-GABAB receptor antagonist that decreases GABA-induced IP3 (inositol trisphosphate) production with an IC50 of 37.9 ?M. It is a selective and negative allosteric modulator of GABAB (?-Aminobutyric acid) receptors.