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View larger Cort108297
AT15000
CAS 1018679-79-2
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $209.10 | Total: $1,045.50 |
| 1 | 10 | $177.12 | Total: $1,771.20 |
| 1 | 25 | $150.06 | Total: $3,751.50 |
| 1 | 50 | $127.92 | Total: $6,396.00 |
| 1 | 100 | $110.70 | Total: $11,070.00 |
Data sheet
| Molecular Formula | C26H25F4N3O3S |
| Molecular Weight | 535.55 |
| CAS Numbers | 1018679-79-2 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCOC[C@@]12CN(CCC1=Cc1c(C2)cnn1-c1ccc(F)cc1)S(=O)(=O)c1ccc(cc1)C(F)(F)F |
| References | Sindelar DK, et al. LLY-2707, a novel nonsteroidal glucocorticoid antagonist that reduces atypical antipsychotic-associated weight gain in rats. J Pharmacol Exp Ther. 2014 Jan;348[1] 192-201. |
More info
Cort108297 is a selective glucocorticoid receptor modulator and a selective GR antagonist with no affinity for other steroid receptors. Cort108297 showed a high affinity for GRs (Ki: 0.45nM).