Histamine Receptors

Ritanserin View larger

Ritanserin

AT16759

CAS 87051-43-2

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$29.00

$29.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $13.05 Total: $1,305.00
150 $15.08 Total: $754.00
125 $17.69 Total: $442.25
110 $20.88 Total: $208.80
15 $24.65 Total: $123.25

Data sheet

Molecular FormulaC27H25F2N3OS
Molecular Weight477.57
CAS Numbers87051-43-2
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCc1nc2sccn2c(=O)c1CCN1CCC(CC1)=C(c1ccc(F)cc1)c1ccc(F)cc1
ReferencesLeysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27[6] 600-11.

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Ritanserin (R 55667) is a highly effective, relatively selective, long-acting 5-HT2 receptor antagonist (IC50: 0.9 nM), with less activity on Histamine H1, Dopamine D2, Adrenergic ?1, and Adrenergic ?2 receptors.