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View larger Samelisant
AT9770
CAS 1394808-82-2
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $81.60 | Total: $408.00 |
| 1 | 10 | $69.12 | Total: $691.20 |
| 1 | 25 | $58.56 | Total: $1,464.00 |
| 1 | 50 | $49.92 | Total: $2,496.00 |
| 1 | 100 | $43.20 | Total: $4,320.00 |
Data sheet
| Molecular Formula | C21H31N3O3 |
| Molecular Weight | 373.49 |
| CAS Numbers | 1394808-82-2 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O(C1CCN(CC1)C2CCC2)C3=CC=C(NC(CN4CCOCC4)=O)C=C3 |
| References | Nirogi R, et al. Samelisant [SUVN-G3031], a potent, selective and orally active histamine H3 receptor inverse agonist for the potential treatment of narcolepsy pharmacological and neurochemical characterisation. Psychopharmacology [Berl]. 2021 Jun;238[6] 1495-1511. |
More info
Samelisant (SUVN-G3031) is a selective and inverse agonist of H3 receptor with Kis of 8.7 nM and 9.8 nM for human and rat. Samelisant has anticataplectic effects and can be used in studies about narcolepsy.